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Click to edit Master title style,Click to edit Master text styles,Second level,Third level,Fourth level,Fifth level,*,先正达(中国)投资有限公司,技术部 叶承道,三唑类杀菌剂竞争分析,甾醇生物合成抑制剂作用方式研究概况,1974 抑制蛋白质合成,1975 抑制生物氧化作用,1980 抑制甾醇合成,1980 麦角甾醇,8,-,7,异构化作用,1981 麦角甾醇,14,-还原作用,1981 麦角甾醇 C,14,-脱甲基作用,麦角甾醇生物合成抑制剂,(EMIs),羊毛甾醇,麦角甾醇,2,4,亚甲基羊毛甾醇,4,4,二甲基麦角甾-8,4,24三烯醇,粪甾醇,4,4,二甲基粪甾醇,14,还原反应,8,7,双键异构化反应,真菌细胞膜,x,x,x,C,14,-,脱甲基反应,14(15)还原酶/8(7)异构酶抑制剂,A,吗啉类(Morpholines),R1=C,12,H,25,(dodemorph),十二环吗啉(1965),BASF,O N,R,R2=C,13,H,27,(tridemorph),十三吗啉(1965),BASF,R3=C,3,H,7,-C,6,H,5,-C,4,H9,(fenpropimorph),丁苯吗啉 (1979),BASF,烯酰吗啉,安克(dimethomorph)-(1984)Rohm&Hass,丁苯吗啉(fenpropimorph)杀菌谱,14(15)还原酶/8(7)异构酶抑制剂,B,哌啶类(Piperidines),C N R,fenpropidin(Patrol),丁苯哌啶(1979),Roche-Maag,甾醇C,14,a,-脱甲基酶抑制剂,(DMIs),A,嘧啶类(Pyrimidines),N C Y,C C C OH,N C X,X=H,Y=Cl 苯嘧啶醇(triarimol,Elacocide)1975 Eli Liiiy/Dow,X=Cl,Y=H 氯 苯嘧啶醇(fenarimol,Rubigan)1976 Eli Lilly/Dow,X=F,Y=H 氟 苯嘧啶醇(nuarimol)1976 Eli Lilly/Dow,A,嘧啶类(Pyrimidines)杀菌谱 乐必耕(fenarimol,Rubigan 氯苯嘧啶醇),B,吡啶类(Pyridines),C C Cl,C C C OH,N C Cl,帕里醇(Parinol)1976 Eli Lilly/Dow,C,咪,咪,唑,唑,类,类(Imidazoles),CC,N,R,NC,OC,3,H,5,R,=,CH,2,CH,Cl,lC,抑,霉,霉,唑,唑(imazalil,Fungflor,万,万,得,得,利,利)1972Janssen,C,咪,咪,唑,唑,类,类(Imidazoles),Cl,OC,2,H,4,OCl,R=CNCl,C,3,H,7,咪,鲜,鲜,胺,胺(prochloraze,Sportak,施,施,保,保,克,克)1977,Schering/Aventis,CF,NCl,R=C,CH,2,OC,3,H,7,氟,菌,菌,唑,唑(triflumizole,Trifumine,特,特,富,富,灵,灵)1979,NipponSoda,C,咪,咪,唑,唑,类,类(Imidazoles),杀,杀,菌,菌,谱,谱,施,施,保,保,克,克(prochloraz,Sportak,咪,咪,鲜,鲜,胺,胺),D,1,三,三,唑,唑,类,类(Triazoles),CN,NR1,NC,R1=CCF,3,三,氟,氟,苯,苯,唑,唑(fluotrimazole,Persalon,氟,氟,霉,霉,唑,唑)1973,Bayer,D,2,三,三,唑,唑,类,类(Triazoles),CN,NCHOCl(R),NCCC(CH,3,),3,O,三,唑,唑,酮,酮(Triadimefon,Bayleton,粉,粉,锈,锈,宁,宁)1972,Bayer,CN,NCHOCl(R),NC,CHC(CH,3,),3,HO,三,唑,唑,醇,醇(triadiminol,Baytan,)1972,Bayer,D,2,三,三,唑,唑,类,类(Triazoles),杀,杀,菌,菌,谱,谱,三,三,唑,唑,酮,酮(tridimifon),D,2,三,三,唑,唑,类,类(Triazoles),R=双,苯,苯,三,三,唑,唑,醇,醇(bitertanol)1981,Bayer,Cl,R=ClCH,2,苄,氯,氯,三,三,唑,唑,醇,醇(diclobutrazole)1981,ICI/Zeneca/Syngenta,*,多,多,效,效,唑,唑(Paclobutrazol,PP333)1981,Cl,R=ClCH,烯,唑,唑,醇,醇(diniconazole,Spotless,速,速,保,保,利,利)1982,Sumitomo,*,烯,烯,效,效,唑,唑(uniconazol,Sumagic)1982,D,3,三,三,唑,唑,类,类(Triazoles),CNOH,NCH2CR2,NCR1,R1=ClC,2,H,4,R2=(CH,3,),3,C,戊,唑,唑,醇,醇(tebuconazole,Raxil,立,立,克,克,秀,秀,Folicur)1981,Bayer,F,R1=F,R2=,粉,唑,唑,醇,醇(flutriafol,Imapact)1983,ICI/Zeneca/Syngenta,Cl,R1=Cl,R2=nC,4,H,9,己,唑,唑,醇,醇(hexaconazole,Anil,安,安,福,福)1985,ICI/Zeneca/Syngenta,D,3,三,三,唑,唑,类,类(Triazoles),杀,杀,菌,菌,谱,谱,立,立,克,克,秀,秀(tebuconazol,Raxil,Folicur,戊,戊,唑,唑,醇,醇),D,3,三,三,唑,唑,类,类(Triazoles),杀,杀,菌,菌,谱,谱,安,安,福,福(hexaconazole,Anvil,己,己,唑,唑,醇,醇),D,4,三,三,唑,唑,类,类(Triazoles),CNCN,NCH2CR2,NCR1,R1=,R2=nC,4,H,9,咪,菌,菌,腈,腈(fenapanil,Sisthan)1976,Rohm-Haas,R1=Cl,R2=nC,4,H,9,腈,菌,菌,唑,唑(myclobutanil,Systhane,仙,仙,生,生)1981,Rohm-Hass,R1=,R2=CF,3,C,2,H,4,唑,菌,菌,腈,腈(propanenitrile,RH7592)1988,Rohm-Hass,D,5,三,三,唑,唑,类,类(Triazoles),杀,杀,菌,菌,谱,谱,仙,仙,生,生(Myclobutanil,Systane,腈,腈,菌,菌,唑,唑),D5,三,三,唑,唑,类,类(Triazoles),Cl,CN,NCH,2,CR2,NCOO,CCR,1,R,1,=CH,3,-,甲,甲,环,环,唑,唑1978,Ciba/Novartis/Syngenta,R,1,=C,2,H,5,-,乙,乙,环,环,唑,唑(etaconazole)1978,Ciba/Novartis/Syngenta,R,1,=n-C,3,H,7,丙,环,环,唑,唑(propiconazole,Tilt)1979,Ciba/Novartis/Syngenta,Cl,R,1,=CH,3,-,R2=-C-O-Cl,苯醚,甲,甲,环,环唑(difenoconazole,Score,世,世,高,高)1983,Ciba/Novartis/Syngenta,D5,三,三唑,类,类(Triazoles),杀,杀菌,谱,谱,敌,敌,力,力脱(propiconazole,Tilt,丙,丙环,唑,唑),D5,三,三唑,类,类(Triazoles),杀,杀菌,谱,谱,世,世,高,高(difenoconazole,Score),D5,世,世高(Score),对,对,蔬,蔬菜,白,白粉,病,病(Erysiphe,白,白粉,菌,菌)(Sphaerotheca,单,单丝,壳,壳菌)和(Leveillula鞑,靼,靼内,丝,丝菌)的,效,效果,D5,世,世高(Score),对,对,蔬,蔬菜,黑,黑斑,病,病(Alternaria,链,链,格,格孢,菌,菌),的,的效,果,果,D5,世,世高(Score),对,对,蔬,蔬菜,褐,褐斑,病,病(Cercospora,尾,尾,孢,孢菌)和,斑,斑枯,病,病(Septoria,壳,壳,针,针孢,菌,菌),的,的效,果,果,D6,三,三唑,类,类(Triazoles),CNCH3,N,CH2SiF,NC,F,氟硅,唑,唑(flusilazole,Nustar,福,福星)1984,DuPont,D6,福,福星(flusilazole,Nustar)杀,菌,菌谱,D7,三,三唑,类,类(Triazoles),环氧,菌,菌唑(epoxiconazole,Opus)75-125gai/ha-1986,BASF,氟喹,唑,唑(fluquinconazole,Casteller)100-200gai/ha,-1986,Rhone-poulenc/Aventis,氟醚,唑,唑(tetraconazole,Arpege)50-100gai/ha-1987,AgrimartCo.,羟菌,唑,唑(metconazole)30-90gai/ha-1987,日,日,本,本吴,羽,羽,呋菌,唑,唑(furconacole)50-100gai/ha-1987,Rhone-poulenc/Aventis,糠菌,唑,唑(bromuconazole)20-30gai/ha,1988,Rhone-poulenc/Aventis,内吸,传,传导,,,,杀,菌,菌谱,广,广,耐雨,冲,冲刷,,,,药,效,效持,久,久,剂型,先,先进,,,,作,物,物安,全,全,低毒,低,低残,,,,环,境,境友,善,善,世高(difenoconazole,Score),特,特点,演讲,完,完毕,,,,谢,谢,谢观,看,看!,
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